What drugs target rho kinase?

2+ drugs target rho kinase, including Rhopressa.

What drug classes act on rho kinase?

Drug classes acting on rho kinase include Rho Kinase Inhibitor, Rho kinase inhibitor.

rho kinase — Drug Target

Name: Drug Landscape Pharmaceutical Database
Creator: Drug Landscape
Published: 2026-01-01
License: https://creativecommons.org/licenses/by/4.0/

2 drugs 1 marketed

All drugs that target rho kinase — marketed and clinical-stage. Includes 2 drug classes acting on this target.

Drug classes

Rho Kinase Inhibitor · Rho kinase inhibitor

Marketed (1)

Rhopressa · Alcon Labs Inc · Rho Kinase Inhibitor · Cardiovascular
Netarsudil reduces intraocular pressure by increasing aqueous humor outflow through the trabecular meshwork.

Phase 2 pipeline (1)

Losmapimod tablets · GlaxoSmithKline · Rho kinase inhibitor · Cardiovascular
Rho kinase inhibitor