What drugs target PD-1 and PD-L1?

1+ drugs target PD-1 and PD-L1, including .

What drug classes act on PD-1 and PD-L1?

Drug classes acting on PD-1 and PD-L1 include PD-1/PD-L1 inhibitor.

PD-1 and PD-L1 — Drug Target

Name: Drug Landscape Pharmaceutical Database
Creator: Drug Landscape
Published: 2026-01-01
License: https://creativecommons.org/licenses/by/4.0/

1 drugs 1 in Phase 3

All drugs that target PD-1 and PD-L1 — marketed and clinical-stage. Includes 1 drug classes acting on this target.

Drug classes

PD-1/PD-L1 inhibitor

Phase 3 pipeline (1)

Full course of PD-1/PD-L1 blockades · Sun Yat-sen University · PD-1/PD-L1 inhibitor · Oncology
PD-1/PD-L1 blockade releases the brakes on the immune system by inhibiting checkpoint proteins that cancer cells use to evade T-cell attack, thereby restoring anti-tumor immunity.