Muscarinic M3 receptor and beta-3 adrenergic receptor — Drug Target
All drugs that target Muscarinic M3 receptor and beta-3 adrenergic receptor — marketed and clinical-stage. Includes 1 drug classes acting on this target.
Drug classes
Antimuscarinic and beta-3 adrenergic agonist combination
Marketed (1)
- tolterodine , mirabegron · Far Eastern Memorial Hospital · Antimuscarinic and beta-3 adrenergic agonist combination · Urology
Tolterodine and mirabegron work together to reduce overactive bladder symptoms through complementary pathways: tolterodine blocks muscarinic receptors to decrease bladder contractions, while mirabegron activates beta-3 adrenergic receptors to relax the detrusor muscle.