bradykinin B2 receptor — Drug Target
All drugs that target bradykinin B2 receptor — marketed and clinical-stage. Includes 1 drug classes acting on this target.
Drug classes
Bradykinin B2 receptor antagonist
Marketed (1)
- ICATIBANT ACETATE
Icatibant blocks bradykinin from binding to the B2 receptor, reducing HAE symptoms.
Phase 2 pipeline (1)
- HOE140 Icatibant · Sanofi · Bradykinin B2 receptor antagonist · Immunology / Rare Disease
Icatibant is a selective bradykinin B2 receptor antagonist that blocks the inflammatory effects of bradykinin, a key mediator of angioedema.