A2A receptor — Drug Target

All drugs that target A2A receptor — marketed and clinical-stage. Includes 4 drug classes acting on this target.

Drug classes

A2A receptor agonist · Adenosine receptor agonist · adenosine receptor agonist · adenosine A2A receptor antagonist

Phase 3 pipeline (3)

• Regadenoson central -central · Lokien van Nunen · A2A receptor agonist · Cardiovascular
  Regadenoson central acts as an adenosine A2A receptor agonist, increasing coronary blood flow.
• Regadenoson central - peripheral · Lokien van Nunen · Adenosine receptor agonist · Cardiovascular
  Regadenoson central - peripheral acts as an adenosine A2A receptor agonist.
• Regadenoson; Optison · University of Nebraska · adenosine receptor agonist · Cardiovascular
  Regadenoson is a selective adenosine A2A receptor agonist.

Phase 2 pipeline (2)

• AZD5148 · AstraZeneca · adenosine A2A receptor antagonist · Oncology
  AZD5148 is a selective, potent and orally bioavailable adenosine A2A receptor antagonist.
• AZD8529 · AstraZeneca · adenosine A2A receptor antagonist · Oncology
  AZD8529 is a selective adenosine A2A receptor antagonist.