US Patent

US9820985 — Dihydropyridophthalazinone inhibitors of poly(ADP-ribose)polymerase (PARP)

Method of Use · Assigned to Medivation Technologies LLC · Expires 2029-07-27 · 3y remaining

Vulnerability score 81/100 Vulnerable — likely target for IPR or design-around

What this patent protects

This patent protects pharmaceutical compositions that inhibit poly(ADP-ribose)polymerase activity and their use in treating diseases, disorders, and conditions.

USPTO Abstract

A compound having the structure set forth in Formula (I) and Formula (II): wherein the substituents Y, Z, A, B, R 1 , R 2 , R 3 , R 4 and R 5 are as defined herein. Provided herein are inhibitors of poly(ADP-ribose)polymerase activity. Also described herein are pharmaceutical compositions that include at least one compound described herein and the use of a compound or pharmaceutical composition described herein to treat diseases, disorders and conditions that are ameliorated by the inhibition of PARP activity.

Drugs covered by this patent

FDA Patent Use Codes

When a patent is method-of-use, FDA lists it once per applicable indication ("U-code"). Each U-code carves out a specific therapeutic use that generic filers must either license or design around.

CodeDescriptionDrug
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna
U-2437 Talzenna

Patent Metadata

Patent number
US9820985
Jurisdiction
US
Classification
Method of Use
Expires
2029-07-27
Drug substance claim
No
Drug product claim
No
Assignee
Medivation Technologies LLC
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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