US Patent

US9732075 — Benzimidazole-proline derivatives

Method of Use · Assigned to Idorsia Pharmaceuticals Ltd · Expires 2033-06-12 · 7y remaining

Vulnerability score 53/100 Moderate — design-around opportunities exist

What this patent protects

This patent protects benzimidazole-proline derivatives, specifically compounds of formula (I), and their use as orexin receptor antagonists.

USPTO Abstract

The present invention relates to compounds of the formula (I) wherein Ar 1 , R 1 , R 2 , R 3 , R 4a , R 4b and (R 5 ) n are as described in the description, to their preparation, to pharmaceutically acceptable salts thereof, and to their use as pharmaceuticals, to pharmaceutical compositions containing one or more compounds of formula (I), and especially to their use as orexin receptor antagonists.

Drugs covered by this patent

FDA Patent Use Codes

When a patent is method-of-use, FDA lists it once per applicable indication ("U-code"). Each U-code carves out a specific therapeutic use that generic filers must either license or design around.

CodeDescriptionDrug
U-620 daridorexant-hydrochloride
U-620 daridorexant-hydrochloride

Patent Metadata

Patent number
US9732075
Jurisdiction
US
Classification
Method of Use
Expires
2033-06-12
Drug substance claim
Yes
Drug product claim
Yes
Assignee
Idorsia Pharmaceuticals Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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