US Patent
US7504509 — Compounds and methods for development of Ret modulators
Composition of Matter · Assigned to Plexxikon Inc · Expires 2026-10-22 · 0y remaining
Vulnerability score
27/100
Strong — defensible against typical IPR challenges
What this patent protects
This patent protects compounds that modulate the Ret protein and methods for developing such compounds, including crystal structures of Ret surrogates.
USPTO Abstract
Compounds active on Ret are described, as well as methods of using such compounds. Also described are crystal structures of Ret surrogates that were determined using X-ray crystallography. The use of such Ret surrogate crystals and structural information can, for example, be used for identifying molecular scaffolds and for developing ligands that bind to and modulate Ret and for identifying improved ligands based on known ligands.
Drugs covered by this patent
- Zelboraf (vemurafenib) · Hoffmann La Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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