US Patent

US7049320 — NK1 antagonists

Method of Use · Assigned to Schering Corp · Expires 2028-08-19 · 2y remaining

Vulnerability score 75/100 Vulnerable — likely target for IPR or design-around

What this patent protects

This patent protects a NK1 antagonist, specifically a compound with a certain formula, useful for treating various disorders and conditions.

USPTO Abstract

A NK 1 antagonist having the formula (I), wherein Ar 1 and Ar 2 are optionally substituted phenyl or heteroaryl, X 1 is an ether, thio or imino linkage, R 4 and R 5 are not both H or alkyl, and the remaining variables are as defined in the specification, useful for treating a number of disorders, including emesis, depression, anxiety and cough. Pharmaceutical compositions. Methods of treatment and combinations with other agents are also disclosed.

Drugs covered by this patent

FDA Patent Use Codes

When a patent is method-of-use, FDA lists it once per applicable indication ("U-code"). Each U-code carves out a specific therapeutic use that generic filers must either license or design around.

CodeDescriptionDrug
U-1741 rolapitant-hydrochloride
U-1741 rolapitant-hydrochloride

Patent Metadata

Patent number
US7049320
Jurisdiction
US
Classification
Method of Use
Expires
2028-08-19
Drug substance claim
Yes
Drug product claim
Yes
Assignee
Schering Corp
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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