US Patent

US12564590 — Combinations of menin inhibitors and CYP3A4 inhibitors and methods of use thereof

Method of Use · Assigned to Syndax Pharmaceuticals Inc · Expires 2042-12-18 · 17y remaining

Vulnerability score 75/100 Vulnerable — likely target for IPR or design-around

What this patent protects

This patent protects combinations of menin inhibitors with CYP3A4 inhibitors for treating cancer and other diseases.

USPTO Abstract

The present invention is directed to combinations of menin inhibitors with one or more CYP3A4 inhibitors, pharmaceutical compositions thereof, and methods of treating cancer and other diseases mediated by the menin-HLL interaction. Accordingly, the present disclosure provides compounds, e.g., of Formula (II), which inhibit menin and are useful in the treatment of diseases mediated by the menin-MLL interaction in combination with a strong CYP3A4 inhibitor.

Drugs covered by this patent

FDA Patent Use Codes

When a patent is method-of-use, FDA lists it once per applicable indication ("U-code"). Each U-code carves out a specific therapeutic use that generic filers must either license or design around.

CodeDescriptionDrug
U-4045 revumenib-citrate
U-4327 revumenib-citrate
U-4327 revumenib-citrate

Patent Metadata

Patent number
US12564590
Jurisdiction
US
Classification
Method of Use
Expires
2042-12-18
Drug substance claim
No
Drug product claim
Yes
Assignee
Syndax Pharmaceuticals Inc
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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