US Patent
US12491164 — Muco-adhesive, controlled release formulation of levodopa and/or esters of levodopa and uses thereof
Formulation · Assigned to Impax Laboratories LLC · Expires 2034-10-07 · 8y remaining
Vulnerability score
38/100
Strong — defensible against typical IPR challenges
What this patent protects
This patent protects a muco-adhesive, controlled release oral solid formulation of levodopa and/or esters of levodopa with carbidopa.
USPTO Abstract
The invention provides an oral solid formulation comprising (a) a plurality of controlled release components comprising (i) a core comprising a mixture of levodopa and at least one pharmaceutically acceptable excipient, (ii) a controlled release coating surrounding the core, (iii) a muco-adhesive coating surrounding the controlled release coating and (iv) an enteric coating surrounding the muco-adhesive coating; and (b) one or more immediate release components comprising levodopa. The oral solid formulation also contains carbidopa and about 80% to 100% of the carbidopa in the oral solid formulation is present in the one or more immediate release components.
Drugs covered by this patent
- Sinemet Cr (CARBIDOPA) · Aton
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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