US Patent

US12187739 — Diaryl macrocycle polymorph

Formulation · Assigned to Turning Point Therapeutics Inc · Expires 2036-07-05 · 10y remaining

Vulnerability score 55/100 Moderate — design-around opportunities exist

What this patent protects

This patent protects polymorphs of a specific compound useful in treating diseases like cancer in mammals, including humans.

USPTO Abstract

This disclosure relates to polymorphs of (7S,13R)-11-fluoro-7,13-dimethyl-6,7,13,14-tetrahydro-1,15-ethenopyrazolo[4,3-f][1,4,8,10]benzoxatriazacyclotridecin-4(5H)-one that are useful in the treatment of disease, such as cancer, in mammals. This disclosure also relates to compositions including such polymorphs, and to methods of using such compositions in the treatment of diseases, such as cancer, in mammals, especially in humans.

Drugs covered by this patent

Patent Metadata

Patent number
US12187739
Jurisdiction
US
Classification
Formulation
Expires
2036-07-05
Drug substance claim
No
Drug product claim
Yes
Assignee
Turning Point Therapeutics Inc
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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