US Patent
US11795178 — Compositions of thienopyrimidine derivatives
Composition of Matter · Assigned to Takeda Pharmaceutical Co Ltd · Expires 2033-09-27 · 7y remaining
Vulnerability score
0/100
Ironclad — strong claim type, well-established, deep family
What this patent protects
This patent protects a method for producing a thienopyrimidine derivative with gonadotropin releasing hormone antagonistic action.
USPTO Abstract
The present invention provides a production method of a thienopyrimidine derivative or a salt thereof which has a gonadotropin releasing hormone (GnRH) antagonistic action with high quality in high yield. The present invention provides a method of producing a thienopyrirnidine derivative, which comprises reacting 6-(4-aminophenyl)-1-(2,6-difluorobenzyl)-5-dimethylaminomethyl-3-(6-methoxypyridazin-3-yl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione or salt thereof, 1,1â²-carbonyldiimidazole or a salt thereof and methoxyamine or a salt thereof, and the like.
Drugs covered by this patent
- Estrace (ESTRADIOL) · Pfizer
- Orgovyx (relugolix) · MYOVANT SCIENCES
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.