US Patent

US11608343 — Substituted pyrimido[5,4-d]pyrimidines as HER2 inhibitors

Method of Use · Assigned to Boehringer Ingelheim International GmbH · Expires 2041-07-21 · 15y remaining

Vulnerability score 75/100 Vulnerable — likely target for IPR or design-around

What this patent protects

This patent protects new compounds and their use as inhibitors of the HER2 protein and its mutants in treating and preventing oncological diseases.

USPTO Abstract

The present invention relates to new [1,3]diazino[5,4-d]pyrimidines and derivatives of Formula (I) wherein the groups R 1 , R 2 , R 3 and R 4 have the meanings given in the claims and specification, their use as inhibitors of HER2 and its mutants, pharmaceutical compositions which contain such compounds and their use as medicaments, especially as agents for treatment and/or prevention of oncological diseases.

Drugs covered by this patent

FDA Patent Use Codes

When a patent is method-of-use, FDA lists it once per applicable indication ("U-code"). Each U-code carves out a specific therapeutic use that generic filers must either license or design around.

CodeDescriptionDrug
U-4245 Hernexeos

Patent Metadata

Patent number
US11608343
Jurisdiction
US
Classification
Method of Use
Expires
2041-07-21
Drug substance claim
Yes
Drug product claim
Yes
Assignee
Boehringer Ingelheim International GmbH
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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