US Patent

US11433076 — Preparation containing tetracyclic compound at high dose

Formulation · Assigned to Chugai Pharmaceutical Co Ltd · Expires 2035-04-24 · 9y remaining

Vulnerability score 50/100 Moderate — design-around opportunities exist

What this patent protects

This patent protects an improved solubility of a pharmaceutical composition containing a tetracyclic compound, achieved by forming granules of the compound with a disintegrating agent.

USPTO Abstract

An improved solubility of a pharmaceutical composition or formulation containing a large amount of 9-ethyl-6,6-dimethyl-8-(4-morpholin-4-yl-piperidin-1-yl)-11-oxo-6,11-dihydro-5H-benzo[b]carbazole-3-carbonitrile or a salt thereof can be achieved by forming granules of the compound or salt thereof and allowing the granules to be present together with a disintegrating agent.

Drugs covered by this patent

Patent Metadata

Patent number
US11433076
Jurisdiction
US
Classification
Formulation
Expires
2035-04-24
Drug substance claim
No
Drug product claim
Yes
Assignee
Chugai Pharmaceutical Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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