EP1042325B1 — Nitrogen-containing heterocyclic compounds, their production and use
Assigned to Takeda Pharmaceutical Co Ltd · Expires 2005-09-21 · 21y expired
What this patent protects
A compound of the formula: wherein one of A and D is N and the other is C, or both are N; B is N or C; m is 0-3; R<SUP>1</SUP>, R<SUP>2 </SUP>and R<SUP>3 </SUP>each is (i) H or (ii) a group bound via C, N, O or S; R<SUP>4 </SUP>is a…
USPTO Abstract
A compound of the formula: wherein one of A and D is N and the other is C, or both are N; B is N or C; m is 0-3; R<SUP>1</SUP>, R<SUP>2 </SUP>and R<SUP>3 </SUP>each is (i) H or (ii) a group bound via C, N, O or S; R<SUP>4 </SUP>is a group bound via C; R<SUP>5 </SUP>is H or a group bound via C or O; R<SUP>6 </SUP>is H or a group bound via C; R<SUP>7 </SUP>is a homo- or hetero-cyclic group which may be substituted; or a salt thereof possesses excellent gonadotropin-releasing hormone antagonizing activity, and is useful as a prophylactic or therapeutic agent for sex hormone-dependent diseases, and so forth.
Drugs covered by this patent
- Orgovyx (relugolix) · MYOVANT SCIENCES
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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