EP0544445A2 — Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists
Assigned to Syngenta Ltd · Expires 1993-06-02 · 33y expired
What this patent protects
Compounds of formula I, and pharmaceutically acceptable salts thereof, in which R1 is hydrogen (1-6C)alkyl or (1-4C)alkanoyl ; A is -N=CQ-O-, N=CQ-NR 8 -, -N=CQ-CH=Nor -N=CH-CQ=N- ; Q is 2-furyl ; R 8 is hydrogen or C1-4C)alkyl ; and R 2 has any of the mea…
USPTO Abstract
Compounds of formula I, and pharmaceutically acceptable salts thereof, in which R1 is hydrogen (1-6C)alkyl or (1-4C)alkanoyl ; A is -N=CQ-O-, N=CQ-NR 8 -, -N=CQ-CH=Nor -N=CH-CQ=N- ; Q is 2-furyl ; R 8 is hydrogen or C1-4C)alkyl ; and R 2 has any of the meanings given in the specification, processes for preparing the compounds and pharmaceutical compositions containing them. The compounds are useful as adenosine antagonists.
Drugs covered by this patent
- Balversa (ERDAFITINIB) · Johnson & Johnson
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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