EP0251315A2 — Naphthalene derivatives, process for their preparation and pharmaceutical compositions containing the same
Assigned to Tanabe Pharma Corp · Expires 1988-01-07 · 38y expired
What this patent protects
Naphthalene derivative of the formula: wherein Ring A is a substituted or unsubstituted benzene ring; each of R¹ and R² is a group of the formula: -OR⁵, -NHR⁵ or ; or either one of R¹ and R² is a lower alkoxy group and other one is a group of the formula: -OR⁵, -NHR⁵ …
USPTO Abstract
Naphthalene derivative of the formula: wherein Ring A is a substituted or unsubstituted benzene ring; each of R¹ and R² is a group of the formula: -OR⁵, -NHR⁵ or ; or either one of R¹ and R² is a lower alkoxy group and other one is a group of the formula: -OR⁵, -NHR⁵ or ; each of R³ and R⁴ is a lower alkoxy group, or one of R³ and R⁴ is a lower alkoxy group and the other is a hydrogen atom; R⁵ is a substituted alkyl group, a heterocyclic group, a cycloalkyl group, an alkyl group of at least 5 carbon atoms or alkenyl group; and each of R⁶ and R⁷ is hydrogen atom or a lower alkyl group and salts thereof are disclosed. Said naphthalene derivative (I) and its salts have excellent hypolipidemic activity and are useful for treatment or prophylaxis of hyperlipidemia and/or arteriosclerosis.
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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