EP0009384A1 — Processes for the preparation of triazinones and condensed triazinones, and compounds so obtained
Assigned to Glaxo Group Ltd · Expires 1980-04-02 · 46y expired
What this patent protects
Compounds of the formula (I)(in which X represents HS- or a group R,R<sub>2</sub>N- wherein R, and R<sub>2</sub> which may be the same or different represent hydrogen or a straight or branched chain alkyl group containing from 1 to 4 carbon atoms or a benz…
USPTO Abstract
Compounds of the formula (I)(in which X represents HS- or a group R,R<sub>2</sub>N- wherein R, and R<sub>2</sub> which may be the same or different represent hydrogen or a straight or branched chain alkyl group containing from 1 to 4 carbon atoms or a benzyl group and R<sub>3</sub> represents a C<sub>3-2</sub> alkyl group or a C<sub>3-2</sub> cycloalkyl group) are prepared by reacting an α-ketoester of the formula (II)(in which Alk represents an alkyl group) or a precursor thereof with a compound of the formula (III)The precursor of the compound of formula (II) may be a mixture of isomeric enol estersThe compounds of formula (I) may be converted into compounds of formula (VIII)in which R, and R<sub>2</sub> which may be the same or different represent hydrogen or a straight or branched chain alkyl group containing from 1 to 4 carbon atoms, and R<sub>3</sub> is as defined above.
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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