CN Patent

CN1914191A — 4-(4-甲基哌嗪-1-基甲基)-n-[4-甲基-3-(4-吡啶-3-基)嘧啶-2-基氨基)苯基]-苯甲酰胺的盐形式

Assigned to Novartis AG · Expires 2007-02-14 · 19y expired

What this patent protects

本发明涉及4-[(4-甲基-1-哌嗪基)甲基]-N-[4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯基]-苯甲酰胺的酸加成盐,其选自酒石酸盐,如(D)(-)酒石酸盐或(L)(+)酒石酸盐、盐酸盐、柠檬酸盐、苹果酸盐、富马酸盐、琥珀酸盐、苯甲酸盐、苯磺酸盐、双羟萘酸盐、甲酸盐、丙二酸盐、1,5-萘二磺酸盐、水杨酸盐、环己烷氨基磺酸盐、乳酸盐、扁桃酸盐、含水戊二酸盐、己二酸盐、方酸盐、香草酸盐、草酰乙酸盐、抗坏血酸盐和硫酸盐。

USPTO Abstract

本发明涉及4-[(4-甲基-1-哌嗪基)甲基]-N-[4-甲基-3-[[4-(3-吡啶基)-2-嘧啶基]氨基]苯基]-苯甲酰胺的酸加成盐,其选自酒石酸盐,如(D)(-)酒石酸盐或(L)(+)酒石酸盐、盐酸盐、柠檬酸盐、苹果酸盐、富马酸盐、琥珀酸盐、苯甲酸盐、苯磺酸盐、双羟萘酸盐、甲酸盐、丙二酸盐、1,5-萘二磺酸盐、水杨酸盐、环己烷氨基磺酸盐、乳酸盐、扁桃酸盐、含水戊二酸盐、己二酸盐、方酸盐、香草酸盐、草酰乙酸盐、抗坏血酸盐和硫酸盐。

Drugs covered by this patent

Patent Metadata

Patent number
CN1914191A
Jurisdiction
CN
Classification
Expires
2007-02-14
Drug substance claim
No
Drug product claim
No
Assignee
Novartis AG
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

Track this patent

Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.