CN Patent
CN1668283A — 具有提高的溶出度的药物组合物
Assigned to Transform Pharmaceuticals Inc · Expires 2005-09-14 · 21y expired
What this patent protects
本发明涉及筛选含药物化合物和赋形剂的混合物,以鉴定药物化合物/赋形剂组合延缓固态核化的性质的方法。本发明还涉及通过使在胃液条件下具有低溶解度的药物与重结晶/沉淀延缓剂以及任选的增强剂联合,提高药物的溶解度、溶出度和生物利用度。
USPTO Abstract
本发明涉及筛选含药物化合物和赋形剂的混合物,以鉴定药物化合物/赋形剂组合延缓固态核化的性质的方法。本发明还涉及通过使在胃液条件下具有低溶解度的药物与重结晶/沉淀延缓剂以及任选的增强剂联合,提高药物的溶解度、溶出度和生物利用度。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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