CN Patent
CN1610551A — 用作止痛剂的6-羟基羟吗啡酮的肠胃外给药
Assigned to Endo Pharmaceuticals Inc · Expires 2005-04-27 · 21y expired
What this patent protects
在治疗疼痛的方法中,以足以诱导止痛的量向患者给以6-羟基羟吗啡酮的药物组合物。在一种实施方式中,药物组合物是肠胃外给药的,优选地借助注射和静脉内滴注。为了达到所需的止痛效果,6-羟基羟吗啡酮的血浆水平在治疗期间被提升至至少大约0.05ng/ml。以足以诱导止痛的量给以含有6-羟基羟吗啡酮和一种或多种载体、稀释剂和赋形剂的组合物也涵盖其中。
USPTO Abstract
在治疗疼痛的方法中,以足以诱导止痛的量向患者给以6-羟基羟吗啡酮的药物组合物。在一种实施方式中,药物组合物是肠胃外给药的,优选地借助注射和静脉内滴注。为了达到所需的止痛效果,6-羟基羟吗啡酮的血浆水平在治疗期间被提升至至少大约0.05ng/ml。以足以诱导止痛的量给以含有6-羟基羟吗啡酮和一种或多种载体、稀释剂和赋形剂的组合物也涵盖其中。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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