CN Patent
CN1250370A — 鼻内给药的水悬浮液
Assigned to NICHOLAS BOARD · Expires 2000-04-12 · 26y expired
What this patent protects
人们希望将具有优良抗炎和抗过敏活性的氯替泼诺etabonate制成外用药物,但是当其制成水悬浮液时,容易发生聚集和沉淀。根据本发明,通过将氯替泼诺etabonate和微晶纤维素羧甲基纤维素钠一起制成制剂,成功地制成了具有长期稳定性的悬浮液。此外,所制得的悬浮液具有显著改善了的鼻内保留性以及没有皮肤或粘膜刺激作用。
USPTO Abstract
人们希望将具有优良抗炎和抗过敏活性的氯替泼诺etabonate制成外用药物,但是当其制成水悬浮液时,容易发生聚集和沉淀。根据本发明,通过将氯替泼诺etabonate和微晶纤维素羧甲基纤维素钠一起制成制剂,成功地制成了具有长期稳定性的悬浮液。此外,所制得的悬浮液具有显著改善了的鼻内保留性以及没有皮肤或粘膜刺激作用。
Drugs covered by this patent
- Ozempic (semaglutide) · Novo Nordisk
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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