CN Patent
CN121627532A — 一种奥马环素的制备方法
Assigned to Jiangsu Puxin Pharmaceutical Co ltd · Expires 2026-03-10 · 0y expired
What this patent protects
本发明提供了一种奥马环素的制备方法。具体地,本发明的方法包括如下步骤:在惰性气体存在下,在惰性溶剂中,式III所示的化合物与特戊醛反应,得到奥马环素粗品;吸附树脂纯化:将所述奥马环素粗品通过吸附树脂进行纯化,得到奥马环素纯品。本发明的方法收率高、纯度高,适合工业化生产。
USPTO Abstract
本发明提供了一种奥马环素的制备方法。具体地,本发明的方法包括如下步骤:在惰性气体存在下,在惰性溶剂中,式III所示的化合物与特戊醛反应,得到奥马环素粗品;吸附树脂纯化:将所述奥马环素粗品通过吸附树脂进行纯化,得到奥马环素纯品。本发明的方法收率高、纯度高,适合工业化生产。
Drugs covered by this patent
- Nuzyra (OMADACYCLINE TOSYLATE) · Paratek Pharms
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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