CN121319053A — 一类带有二乙烯基磷酰基的2-氨基嘧啶类化合物及其应用
Assigned to Institute Of Basic Medicine And Oncology Chinese Academy Of Sciences Preparatory · Expires 2026-01-13 · 0y expired
What this patent protects
本发明公开了一类带有二乙烯基磷酰基的2‑氨基嘧啶类化合物及其应用。具体地,本发明公开了一种如式(I)所示的化合物、其立体异构体、互变异构体、晶型、药学上可接受的盐、水合物、溶剂合物或前药。本发明的化合物是一种EGFR抑制剂,可以用于制备治疗和/或预防与EGFR相关的疾病的药物。
USPTO Abstract
本发明公开了一类带有二乙烯基磷酰基的2‑氨基嘧啶类化合物及其应用。具体地,本发明公开了一种如式(I)所示的化合物、其立体异构体、互变异构体、晶型、药学上可接受的盐、水合物、溶剂合物或前药。本发明的化合物是一种EGFR抑制剂,可以用于制备治疗和/或预防与EGFR相关的疾病的药物。
Drugs covered by this patent
- Alunbrig (brigatinib) · Takeda
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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