CN Patent
CN121194983A — 5'-膦酸酯修饰的核苷类似物及其制备的寡核苷酸
Assigned to Shanghai Bowang Pharmaceutical Co ltd · Expires 2025-12-23 · 0y expired
What this patent protects
涉及可用于5′修饰的核苷类似物以及由它们制备的寡核苷酸,更具体涉及可用于并入到寡核苷酸末端的修饰核苷及其类似物,可以结合到双链寡核苷酸(短干扰RNA)或单链寡核苷酸(例如反义寡核苷酸)中。预期提供的所述寡核苷酸与靶RNA的一部分杂交,从而导致所述靶RNA正常功能的丧失。
USPTO Abstract
涉及可用于5′修饰的核苷类似物以及由它们制备的寡核苷酸,更具体涉及可用于并入到寡核苷酸末端的修饰核苷及其类似物,可以结合到双链寡核苷酸(短干扰RNA)或单链寡核苷酸(例如反义寡核苷酸)中。预期提供的所述寡核苷酸与靶RNA的一部分杂交,从而导致所述靶RNA正常功能的丧失。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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