CN Patent
CN121181479A — 结晶药物产品的制备
Assigned to Orion Oyj · Expires 2025-12-23 · 0y expired
What this patent protects
本发明涉及N‑((S)‑1‑(3‑(3‑氯‑4‑氰基苯基)‑1H‑吡唑‑1‑基)‑丙烷‑2‑基)‑5‑(1‑羟基乙基)‑1H‑吡唑‑3‑甲酰胺(I)的结晶颗粒,其具有在约8至约16m 2 /g、优选约10至约15m 2 /g的范围内的比表面积(SSA),和制备所述颗粒的方法。化合物(I)是强效的雄激素受体(AR)调节剂,其可用作药物、例如治疗前列腺癌的药物。
USPTO Abstract
本发明涉及N‑((S)‑1‑(3‑(3‑氯‑4‑氰基苯基)‑1H‑吡唑‑1‑基)‑丙烷‑2‑基)‑5‑(1‑羟基乙基)‑1H‑吡唑‑3‑甲酰胺(I)的结晶颗粒,其具有在约8至约16m 2 /g、优选约10至约15m 2 /g的范围内的比表面积(SSA),和制备所述颗粒的方法。化合物(I)是强效的雄激素受体(AR)调节剂,其可用作药物、例如治疗前列腺癌的药物。
Drugs covered by this patent
- Nubeqa (darolutamide) · Bayer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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