CN Patent
CN120265291A — 喹唑啉酮化合物的新用途和制剂
Assigned to F Hoffmann La Roche AG · Expires 2025-07-04 · 1y expired
What this patent protects
本发明涉及(3R)‑N‑[2‑氰基‑4‑氟‑3‑(3‑甲基‑4‑氧代‑喹唑啉‑6‑基)氧基‑苯基]‑3‑氟‑吡咯烷‑1‑磺酰胺或其药用盐,其用于局部晚期实体瘤、特别是有脑转移的黑色素瘤的治疗的新用途中。本发明还涉及包含(3R)‑N‑[2‑氰基‑4‑氟‑3‑(3‑甲基‑4‑氧代‑喹唑啉‑6‑基)氧基‑苯基]‑3‑氟‑吡咯烷‑1‑磺酰胺或其药用盐的药物组合物。
USPTO Abstract
本发明涉及(3R)‑N‑[2‑氰基‑4‑氟‑3‑(3‑甲基‑4‑氧代‑喹唑啉‑6‑基)氧基‑苯基]‑3‑氟‑吡咯烷‑1‑磺酰胺或其药用盐,其用于局部晚期实体瘤、特别是有脑转移的黑色素瘤的治疗的新用途中。本发明还涉及包含(3R)‑N‑[2‑氰基‑4‑氟‑3‑(3‑甲基‑4‑氧代‑喹唑啉‑6‑基)氧基‑苯基]‑3‑氟‑吡咯烷‑1‑磺酰胺或其药用盐的药物组合物。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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