CN Patent

CN120058603B — 一种卡博替尼新晶型

Assigned to Lunan Pharmaceutical Group Corp · Expires 2026-04-14 · 0y expired

What this patent protects

本发明属于药物化学的技术领域,具体为卡博替尼新晶型及其制备方法与应用。本发明所提供的新晶型为卡博替尼‑氨基磺酸‑甲醇共晶,其中有一分子卡博替尼、一分子氨基磺酸和一分子甲醇成晶型的基本单元,在稳定性、溶解性等方面均取得了较大的改善,制备方法操作简单,重现性好,适用于工业化生产。

USPTO Abstract

本发明属于药物化学的技术领域,具体为卡博替尼新晶型及其制备方法与应用。本发明所提供的新晶型为卡博替尼‑氨基磺酸‑甲醇共晶,其中有一分子卡博替尼、一分子氨基磺酸和一分子甲醇成晶型的基本单元,在稳定性、溶解性等方面均取得了较大的改善,制备方法操作简单,重现性好,适用于工业化生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN120058603B
Jurisdiction
CN
Classification
Expires
2026-04-14
Drug substance claim
No
Drug product claim
No
Assignee
Lunan Pharmaceutical Group Corp
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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