CN Patent
CN119019375A — 一种瑞司美替罗新晶型及其制备方法
Assigned to Aoruite Pharmaceutical Tianjin Co ltd · Expires 2024-11-26 · 1y expired
What this patent protects
本发明提供了一种瑞司美替罗新晶型,晶型APTI‑I,使用Cu‑Kα辐射,其以2θ角度表示的X射线粉末衍射图谱在5.0°±0.2°、6.3°±0.2°、7.8°±0.2°、12.2°±0.2°、20.0°±0.2°处有特征峰。该晶型易制备、纯度高、稳定性好,水溶媒中溶解度好,适合工业放大生产和制备药物制剂。
USPTO Abstract
本发明提供了一种瑞司美替罗新晶型,晶型APTI‑I,使用Cu‑Kα辐射,其以2θ角度表示的X射线粉末衍射图谱在5.0°±0.2°、6.3°±0.2°、7.8°±0.2°、12.2°±0.2°、20.0°±0.2°处有特征峰。该晶型易制备、纯度高、稳定性好,水溶媒中溶解度好,适合工业放大生产和制备药物制剂。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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