CN Patent
CN117659020A — 一种咪唑并[1,2-b]哒嗪衍生物及其制备方法和用途
Assigned to Suzhou Langrui Biopharmaceutical Co ltd · Expires 2024-03-08 · 2y expired
What this patent protects
本发明公开了一种式Ⅰ所示的咪唑并[1,2‑b]哒嗪衍生物,或其同位素标记化合物、或其光学异构体、几何异构体、互变异构体或异构体混合物、或其药学上可接受的盐、或其前体药、或其代谢物,以及该衍生物的药物组合物。所述式Ⅰ所示的咪唑并[1,2‑b]哒嗪衍生物或药物组合物可以作为TRK激酶抑制剂,用于治疗或预防由TRK或TRK突变介导的疾病或病症。
USPTO Abstract
本发明公开了一种式Ⅰ所示的咪唑并[1,2‑b]哒嗪衍生物,或其同位素标记化合物、或其光学异构体、几何异构体、互变异构体或异构体混合物、或其药学上可接受的盐、或其前体药、或其代谢物,以及该衍生物的药物组合物。所述式Ⅰ所示的咪唑并[1,2‑b]哒嗪衍生物或药物组合物可以作为TRK激酶抑制剂,用于治疗或预防由TRK或TRK突变介导的疾病或病症。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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