CN117530912A — 适合口服给药的鸟苷酸环化酶-c受体激动剂多肽的稳定的固体制剂
Assigned to Ironwood Pharmaceuticals Inc · Expires 2024-02-09 · 2y expired
What this patent protects
本发明涉及适合口服给药的鸟苷酸环化酶‑C受体激动剂多肽的稳定的固体制剂。本文描述了适合口服给药的稳定的利那洛肽固体制剂,也描述了制备这样的制剂的方法。本文所述的制剂包含由氨基酸序列CysCysGluTyrCysCysAsnProAlaCysThrGlyCysTyr组成的多肽(“利那洛肽”)或其药学上可接受的盐。本文所述的利那洛肽制剂是稳定的,且具有对于生产、储存和分配该药物而言足够的贮存期限。
USPTO Abstract
本发明涉及适合口服给药的鸟苷酸环化酶‑C受体激动剂多肽的稳定的固体制剂。本文描述了适合口服给药的稳定的利那洛肽固体制剂,也描述了制备这样的制剂的方法。本文所述的制剂包含由氨基酸序列CysCysGluTyrCysCysAsnProAlaCysThrGlyCysTyr组成的多肽(“利那洛肽”)或其药学上可接受的盐。本文所述的利那洛肽制剂是稳定的,且具有对于生产、储存和分配该药物而言足够的贮存期限。
Drugs covered by this patent
- Trulance (PLECANATIDE) · Salix
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.