CN Patent

CN117447407B — 一种JAK2抑制剂Pacritinib及其中间体的制备方法

Assigned to Daohe Weifang Pharmaceutical Technology Co ltd · Expires 2024-06-11 · 2y expired

What this patent protects

本发明涉及一种JAK2抑制剂Pacritinib及其中间体的制备方法,Pacritinib的制备方法包括如下步骤: (1)中间体G与中间体H于有机溶剂中,在碱、配体、钯催化剂的作用下,反应得到中间体I;(2)中间体I经烯烃复分解反应得到Pacritinib。

USPTO Abstract

本发明涉及一种JAK2抑制剂Pacritinib及其中间体的制备方法,Pacritinib的制备方法包括如下步骤: (1)中间体G与中间体H于有机溶剂中,在碱、配体、钯催化剂的作用下,反应得到中间体I;(2)中间体I经烯烃复分解反应得到Pacritinib。

Drugs covered by this patent

Patent Metadata

Patent number
CN117447407B
Jurisdiction
CN
Classification
Expires
2024-06-11
Drug substance claim
No
Drug product claim
No
Assignee
Daohe Weifang Pharmaceutical Technology Co ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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