CN Patent
CN117222636A — 作为cdk4/6抑制剂的氘代化合物
Assigned to Gan and Lee Pharmaceuticals Co Ltd · Expires 2023-12-12 · 2y expired
What this patent protects
本发明涉及一种作为CDK4/6抑制剂的氘代化合物、其制备方法、含氘代化合物的药物组合物及其用途,相比于未氘代的对照化合物,具有更佳的代谢稳定性和更优异的药代动力学性质,有望降低临床的使用剂量。
USPTO Abstract
本发明涉及一种作为CDK4/6抑制剂的氘代化合物、其制备方法、含氘代化合物的药物组合物及其用途,相比于未氘代的对照化合物,具有更佳的代谢稳定性和更优异的药代动力学性质,有望降低临床的使用剂量。
Drugs covered by this patent
- Verzenio (abemaciclib) · Eli Lilly
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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