CN Patent
CN117164580A — 一种kras g12c抑制剂的制备方法及其中间体
Assigned to Suzhou Zelgen Biopharmaceutical Co Ltd · Expires 2023-12-05 · 2y expired
What this patent protects
本发明公开了一种KRAS G12C抑制剂的制备方法及其中间体。本发明方法工艺路线简洁、高效、低成本、低污染、安全性高、无柱层析纯化操作,制备的目标产物HPLC纯度大于99.0%,产物的ee值大于99.0%。因此,本发明制备方法更适合工业化应用。
USPTO Abstract
本发明公开了一种KRAS G12C抑制剂的制备方法及其中间体。本发明方法工艺路线简洁、高效、低成本、低污染、安全性高、无柱层析纯化操作,制备的目标产物HPLC纯度大于99.0%,产物的ee值大于99.0%。因此,本发明制备方法更适合工业化应用。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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