CN Patent
CN117143077A — 来那替尼马来酸盐及晶形
Assigned to Wyeth LLC · Expires 2023-12-01 · 2y expired
What this patent protects
本发明涉及(E)‑N‑{4‑[3‑氯‑4‑(2‑吡啶基甲氧基)苯胺基]‑3‑氰基‑7‑乙氧基‑6‑喹啉基}‑4‑(二甲基氨基)‑2‑丁烯酰胺的马来酸盐形式,制备结晶马来酸盐形式的方法,和有关的化合物,以及包含它们的药物组合物。所述马来酸盐可用于治疗癌、特别是受表皮生长因子受体家族激酶影响的那些癌。
USPTO Abstract
本发明涉及(E)‑N‑{4‑[3‑氯‑4‑(2‑吡啶基甲氧基)苯胺基]‑3‑氰基‑7‑乙氧基‑6‑喹啉基}‑4‑(二甲基氨基)‑2‑丁烯酰胺的马来酸盐形式,制备结晶马来酸盐形式的方法,和有关的化合物,以及包含它们的药物组合物。所述马来酸盐可用于治疗癌、特别是受表皮生长因子受体家族激酶影响的那些癌。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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