CN Patent
CN116970028A — 大环拟肽类蛋白酶抑制剂及其用途
Assigned to Tencent Technology Shenzhen Co Ltd · Expires 2023-10-31 · 3y expired
What this patent protects
本申请提出了一种化合物,其为式(I)所示化合物或式(I)所示化合物的立体异构体、互变异构体、氮氧化物、溶剂化物、代谢产物、药学上可接受的盐或它的前药,式(I)所示的化合物能够显著抑制Mpro或抑制冠状病毒复制,并且具有很好的代谢稳定性。
USPTO Abstract
本申请提出了一种化合物,其为式(I)所示化合物或式(I)所示化合物的立体异构体、互变异构体、氮氧化物、溶剂化物、代谢产物、药学上可接受的盐或它的前药,式(I)所示的化合物能够显著抑制Mpro或抑制冠状病毒复制,并且具有很好的代谢稳定性。
Drugs covered by this patent
- Paxlovid (Copackaged) (Nirmatrelvir) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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