CN Patent
CN116963734A — 多重酪胺酸激酶抑制剂的结晶盐、其制备方法及用途
Assigned to Mirati Therapeutics Inc · Expires 2023-10-27 · 3y expired
What this patent protects
本发明涉及多重酪胺酸激酶抑制剂的苹果酸盐。特别地,本发明涉及多重酪胺酸激酶抑制剂(S)‑2‑羟基琥珀酸N‑(3‑氟‑4‑((2‑(5‑(((2‑甲氧基乙基)氨基)甲基)吡啶‑2‑基)噻吩并[3,2‑b]吡啶‑7‑基)氧基)苯基)‑N‑(4‑氟苯基)环丙烷‑1,1‑二甲酰胺(1:1)的苹果酸盐的结晶形式、包含该结晶形式的药物组合物、用于制备该结晶形式的方法和该结晶形式的使用方法。
USPTO Abstract
本发明涉及多重酪胺酸激酶抑制剂的苹果酸盐。特别地,本发明涉及多重酪胺酸激酶抑制剂(S)‑2‑羟基琥珀酸N‑(3‑氟‑4‑((2‑(5‑(((2‑甲氧基乙基)氨基)甲基)吡啶‑2‑基)噻吩并[3,2‑b]吡啶‑7‑基)氧基)苯基)‑N‑(4‑氟苯基)环丙烷‑1,1‑二甲酰胺(1:1)的苹果酸盐的结晶形式、包含该结晶形式的药物组合物、用于制备该结晶形式的方法和该结晶形式的使用方法。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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