CN Patent
CN116601151A — Kras g12c抑制剂的晶型
Assigned to Mirati Therapeutics Inc · Expires 2023-08-15 · 3y expired
What this patent protects
本发明涉及KRas G12C抑制剂及其盐的晶型。具体地,本发明涉及KRas G12C抑制剂2‑[(2S)‑4‑[7‑(8‑氯‑1‑萘基)‑2‑[[(2S)‑1‑甲基吡咯烷‑2‑基]甲氧基]‑6,8‑二氢‑5H‑吡啶并[3,4‑d]嘧啶‑4‑基]‑1‑(2‑氟丙‑2‑烯酰基)哌嗪‑2‑基]乙腈的晶型、包含所述晶型的药物组合物、用于制备所述晶型的过程及其使用方法。
USPTO Abstract
本发明涉及KRas G12C抑制剂及其盐的晶型。具体地,本发明涉及KRas G12C抑制剂2‑[(2S)‑4‑[7‑(8‑氯‑1‑萘基)‑2‑[[(2S)‑1‑甲基吡咯烷‑2‑基]甲氧基]‑6,8‑二氢‑5H‑吡啶并[3,4‑d]嘧啶‑4‑基]‑1‑(2‑氟丙‑2‑烯酰基)哌嗪‑2‑基]乙腈的晶型、包含所述晶型的药物组合物、用于制备所述晶型的过程及其使用方法。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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