CN Patent
CN116589451B — 一种6-氧杂螺[4,5]癸烷类化合物的新晶型、用途及其制备方法
Assigned to Chengdu Shuoder Pharmaceutical Co ltd · Expires 2024-07-09 · 2y expired
What this patent protects
本申请涉及药物晶型领域,具体涉及一种(R)‑2‑(9‑(4‑氟苯基)‑6‑氧杂螺[4,5]癸烷‑9‑基)‑N‑(2‑(吡啶‑4‑基)苄基)乙胺二盐酸盐晶型及其制备方法。本发明所得到的式(I)化合物的晶型具备优良的稳定性,并且所用结晶溶剂低毒低残留,适合于大规模生产放大。
USPTO Abstract
本申请涉及药物晶型领域,具体涉及一种(R)‑2‑(9‑(4‑氟苯基)‑6‑氧杂螺[4,5]癸烷‑9‑基)‑N‑(2‑(吡啶‑4‑基)苄基)乙胺二盐酸盐晶型及其制备方法。本发明所得到的式(I)化合物的晶型具备优良的稳定性,并且所用结晶溶剂低毒低残留,适合于大规模生产放大。
Drugs covered by this patent
- Olinvyk (OLICERIDINE) · Trevena
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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