CN Patent
CN116283928A — 一种哒嗪类化合物、其制备方法和应用
Assigned to Ailikang Pharmaceutical Co ltd · Expires 2023-06-23 · 3y expired
What this patent protects
本发明涉及一种如式I所示的一种哒嗪类化合物及其立体异构体、或其药学上可接受的盐、其制备方法、组合物和应用。本发明的Tyk2抑制剂化合物及其异构体、或其药学可接受的盐能够降低Tyk2的酶活性,预防和/或治疗与Tyk2抑制有关的适应症,比如多发性硬化症、类风湿性关节炎、强直性脊柱炎、炎性肠病、系统性红斑狼疮、银屑病、银屑病性关节炎、克罗恩病、舍格伦综合征或硬皮病。
USPTO Abstract
本发明涉及一种如式I所示的一种哒嗪类化合物及其立体异构体、或其药学上可接受的盐、其制备方法、组合物和应用。本发明的Tyk2抑制剂化合物及其异构体、或其药学可接受的盐能够降低Tyk2的酶活性,预防和/或治疗与Tyk2抑制有关的适应症,比如多发性硬化症、类风湿性关节炎、强直性脊柱炎、炎性肠病、系统性红斑狼疮、银屑病、银屑病性关节炎、克罗恩病、舍格伦综合征或硬皮病。
Drugs covered by this patent
- Sotyktu (DEUCRAVACITINIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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