CN Patent
CN116178251A — 一种依度沙班中间体的制备方法
Assigned to Shanghai Huilun Jiangsu Pharmaceutical Co ltd · Expires 2023-05-30 · 3y expired
What this patent protects
本发明提供一种依度沙班中间体的制备方法,所述方法为在有机碱存在下,使化合物式I与化合物式II或其盐进行反应制备得到,在所述反应步骤中单独加入草酸,能够显著提高反应的产率并降低产物中的杂质含量。
USPTO Abstract
本发明提供一种依度沙班中间体的制备方法,所述方法为在有机碱存在下,使化合物式I与化合物式II或其盐进行反应制备得到,在所述反应步骤中单独加入草酸,能够显著提高反应的产率并降低产物中的杂质含量。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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