CN Patent
CN116171155B — 吡啶并[2,3-d]嘧啶-2(1H)-酮衍生物及其制备方法和应用
Assigned to Abbisko Therapeutics Co Ltd · Expires 2024-09-17 · 2y expired
What this patent protects
一种吡啶并[2,3‑d]嘧啶‑2(1H)‑酮衍生物及其制备方法和应用。所述衍生物用于制备治疗至少部分由K‑RAS G12C突变介导的癌症或肿瘤的药物,特别是治疗肺部、肝胆、胃肠道、血液系统、皮肤、骨、泌尿生殖道、神经系统、妇科性和肾上腺相关恶性肿瘤或癌症的药物,有望开发成新一代K‑RAS G12C抑制剂药物。
USPTO Abstract
一种吡啶并[2,3‑d]嘧啶‑2(1H)‑酮衍生物及其制备方法和应用。所述衍生物用于制备治疗至少部分由K‑RAS G12C突变介导的癌症或肿瘤的药物,特别是治疗肺部、肝胆、胃肠道、血液系统、皮肤、骨、泌尿生殖道、神经系统、妇科性和肾上腺相关恶性肿瘤或癌症的药物,有望开发成新一代K‑RAS G12C抑制剂药物。
Drugs covered by this patent
- Lumakras (SOTORASIB) · Amgen
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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