CN Patent
CN115919866A — 特泊替尼固体分散体及其制备方法
Assigned to Shenzhen Neptunus Pharmaceutical Research Institute Co Ltd · Expires 2023-04-07 · 3y expired
What this patent protects
本发明提供了一种特泊替尼固体分散体,该组合物包含水溶性聚合物载体和特泊替尼,二者的所占质量比为5:1~20:1。本发明提供的特泊替尼固体分散体在常温状态下稳定存在,制备过程中工艺参数可控,制备过程简单,能够显著提高特泊替尼的溶解度、改善生物利用度。本发明还提供了一种该特泊替尼固体分散体的制备方法。
USPTO Abstract
本发明提供了一种特泊替尼固体分散体,该组合物包含水溶性聚合物载体和特泊替尼,二者的所占质量比为5:1~20:1。本发明提供的特泊替尼固体分散体在常温状态下稳定存在,制备过程中工艺参数可控,制备过程简单,能够显著提高特泊替尼的溶解度、改善生物利用度。本发明还提供了一种该特泊替尼固体分散体的制备方法。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.