CN Patent

CN115737568A — 一种利培酮鼻用粉雾剂及其制备方法

Assigned to Southeast University · Expires 2023-03-07 · 3y expired

What this patent protects

本发明涉及一种利培酮鼻用粉雾剂及其制备方法,所述制备方法,包括如下步骤:步骤1、将利培酮和增溶剂加入到质量浓度为45‑55%的乙醇溶液中,搅拌溶解均匀,制成喷雾干燥前驱液;步骤2、将喷雾干燥前驱液喷雾干燥,收集粉末,即利培酮鼻用粉雾剂。本发明工艺简单、制剂稳定性好,起效快速,具有较高的可释放剂量,且剂型给药方式简便,相较于传统的口服片剂及注射制剂而言,提高了精神患者的给药依从性。

USPTO Abstract

本发明涉及一种利培酮鼻用粉雾剂及其制备方法,所述制备方法,包括如下步骤:步骤1、将利培酮和增溶剂加入到质量浓度为45‑55%的乙醇溶液中,搅拌溶解均匀,制成喷雾干燥前驱液;步骤2、将喷雾干燥前驱液喷雾干燥,收集粉末,即利培酮鼻用粉雾剂。本发明工艺简单、制剂稳定性好,起效快速,具有较高的可释放剂量,且剂型给药方式简便,相较于传统的口服片剂及注射制剂而言,提高了精神患者的给药依从性。

Drugs covered by this patent

Patent Metadata

Patent number
CN115737568A
Jurisdiction
CN
Classification
Expires
2023-03-07
Drug substance claim
No
Drug product claim
No
Assignee
Southeast University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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