CN Patent
CN115485277A — 作为HER2抑制剂的[1,3]二嗪基[5,4-d]嘧啶
Assigned to Boehringer Ingelheim International GmbH · Expires 2022-12-16 · 3y expired
What this patent protects
本发明涉及式(I)的新的[1,3]二嗪基[5,4‑d]嘧啶及其衍生物,其中基团R 1 、R 2 、R 3 及R 4 具有权利要求书和说明书中所给出的含义;涉及其作为HER2及其突变体的抑制剂的用途;涉及含有此类化合物的药物组合物;及其作为药物,尤其是作为用于治疗和/或预防致癌疾病的药剂的用途。
USPTO Abstract
本发明涉及式(I)的新的[1,3]二嗪基[5,4‑d]嘧啶及其衍生物,其中基团R 1 、R 2 、R 3 及R 4 具有权利要求书和说明书中所给出的含义;涉及其作为HER2及其突变体的抑制剂的用途;涉及含有此类化合物的药物组合物;及其作为药物,尤其是作为用于治疗和/或预防致癌疾病的药剂的用途。
Drugs covered by this patent
- Hernexeos (ZONGERTINIB) · Boehringer Ingelheim
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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