CN Patent
CN115417827B — 6-氨基-1,3,5-三嗪类化合物及其合成方法和应用
Assigned to China Pharmaceutical University · Expires 2023-05-26 · 3y expired
What this patent protects
本发明公开了一种6‑氨基‑1,3,5‑三嗪类化合物或其可药用的盐,化合物结构如通式(I)所示。所述化合物对BTK均有较强的抑制作用,同时能够拮抗肿瘤细胞Raji、Ramos增殖,通过选择性与BTK的不可逆结合并抑制其活性,阻断BCR信号通路,对淋巴瘤有较好的抑制作用。
USPTO Abstract
本发明公开了一种6‑氨基‑1,3,5‑三嗪类化合物或其可药用的盐,化合物结构如通式(I)所示。所述化合物对BTK均有较强的抑制作用,同时能够拮抗肿瘤细胞Raji、Ramos增殖,通过选择性与BTK的不可逆结合并抑制其活性,阻断BCR信号通路,对淋巴瘤有较好的抑制作用。
Drugs covered by this patent
- Imbruvica (ibrutinib) · AbbVie
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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