CN Patent
CN115385899B — ROCK2抑制剂belumosudil的氘代药物及用途
Assigned to Yaokang Zhongtuo Jiangsu Pharmaceutical Technology Co ltd · Expires 2024-04-02 · 2y expired
What this patent protects
本发明公开了ROCK2抑制剂belumosudil的氘代化合物及其药学上可接受的盐,如下式Ⅰ所示,本发明所述的ROCK2抑制剂belumosudil的氘代药物,能进一步降低belumosudil的给药剂量和可能的毒副作用,改善了药代动力学性质。
USPTO Abstract
本发明公开了ROCK2抑制剂belumosudil的氘代化合物及其药学上可接受的盐,如下式Ⅰ所示,本发明所述的ROCK2抑制剂belumosudil的氘代药物,能进一步降低belumosudil的给药剂量和可能的毒副作用,改善了药代动力学性质。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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