CN Patent
CN115385896B — 一种csf-1r抑制剂中间体或其酸式盐的制备方法
Assigned to Abbisko Therapeutics Co Ltd · Expires 2024-11-15 · 2y expired
What this patent protects
本发明涉及一种CSF‑1R抑制剂中间体或其酸式盐的制备方法。所述制备方法以2‑氯‑4‑氟吡啶或其酸式盐为原料,经三步反应制备得到。本发明制备方法原料易得,操作简单,各步收率相对现有技术有很大提高,且工艺稳定,可适应工业化生产需求,解决药物可及性问题,有利于加速CSF‑1R抑制剂的临床开发和药物上市。
USPTO Abstract
本发明涉及一种CSF‑1R抑制剂中间体或其酸式盐的制备方法。所述制备方法以2‑氯‑4‑氟吡啶或其酸式盐为原料,经三步反应制备得到。本发明制备方法原料易得,操作简单,各步收率相对现有技术有很大提高,且工艺稳定,可适应工业化生产需求,解决药物可及性问题,有利于加速CSF‑1R抑制剂的临床开发和药物上市。
Drugs covered by this patent
- Romvimza (VIMSELTINIB) · Deciphera Pharms
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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