CN Patent
CN115215797B — 一种苹果酸卡博替尼新晶型及其制备方法
Assigned to Sichuan Qingmu Pharmaceutical Co ltd · Expires 2024-04-12 · 2y expired
What this patent protects
本发明提供了一种L‑苹果酸卡博替尼新晶型及其制备方法,属于药物晶型领域。针对现有技术中溶解度很低,稳定性较差等问题,本申请开发了一种L‑苹果酸卡博替尼新晶型FormA。该新晶型为L‑苹果酸卡博替尼无水晶型,该晶型相比于现有技术具有在水中溶解度大,稳定性更好等优点,其制备方法简单,环保,重复性好,适合工业放大生产。
USPTO Abstract
本发明提供了一种L‑苹果酸卡博替尼新晶型及其制备方法,属于药物晶型领域。针对现有技术中溶解度很低,稳定性较差等问题,本申请开发了一种L‑苹果酸卡博替尼新晶型FormA。该新晶型为L‑苹果酸卡博替尼无水晶型,该晶型相比于现有技术具有在水中溶解度大,稳定性更好等优点,其制备方法简单,环保,重复性好,适合工业放大生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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